Racemorphan

Racemorphan
Legal status
Legal status	AU: S9 (Prohibited) ; CA: Schedule I ; DE: Anlage II (Authorized trade only, not prescriptible) ; UK: Class A ; US: Schedule II ; UN: Psychotropic Schedule I ;
Identifiers
	IUPAC name (±)-17-Methylmorphinan-3-ol;
CAS Number	297-90-5 ; 5985-35-3 (HBr);
PubChem CID	3918;
ChemSpider	3781;
UNII	V7R79HN3XD;
ChEMBL	CHEMBL20803;
ECHA InfoCard	100.005.499
Chemical and physical data
Formula	C17H23NO
Molar mass	257.37 g/mol
3D model (JSmol)	Interactive image;
	SMILES CN1CCC23CCCCC2C1Cc4ccc(O)cc34;
	InChI InChI=1S/C17H23NO/c1-18-9-8-17-7-3-2-4-14(17)16(18)10-12-5-6-13(19)11-15(12)17/h5-6,11,14,16,19H,2-4,7-10H2,1H3; Key:JAQUASYNZVUNQP-UHFFFAOYSA-N;

Racemorphan, or morphanol, is the racemic mixture of the two stereoisomers of 17-methylmorphinan-3-ol, each with differing pharmacology and effects:

Dextrorphan - an antitussive and dissociative hallucinogen (NMDA receptor antagonist)
Levorphanol - an opioid analgesic

Racemorphan itself is under international control per the Single Convention on Narcotic Drugs 1961 and is therefore listed as a Schedule II Narcotic controlled substance in the US Controlled Substances Act 1970; it has an ACSCN of 9733 and in 2014 it had an aggregate annual manufacturing quota of zero. ^[1] The salts in use are hydrobromide (free base conversion ratio 0.741), hydrochloride (0.876), and tartrate (0.632).

References

↑ "Conversion Factors for Controlled Substances". www.deadiversion.usdoj.gov.

This article is issued from Wikipedia. The text is licensed under Creative Commons - Attribution - Sharealike. Additional terms may apply for the media files.

[1] "Conversion Factors for Controlled Substances". www.deadiversion.usdoj.gov.

Legal status

Legal status	AU: S9 (Prohibited) CA: Schedule I DE: Anlage II (Authorized trade only, not prescriptible) UK: Class A US: Schedule II UN: Psychotropic Schedule I
Identifiers
IUPAC name (±)-17-Methylmorphinan-3-ol
CAS Number	297-90-5 5985-35-3 (HBr)
PubChem CID	3918
ChemSpider	3781
UNII	V7R79HN3XD
ChEMBL	CHEMBL20803
ECHA InfoCard	100.005.499
Chemical and physical data
Formula	C₁₇H₂₃NO
Molar mass	257.37 g/mol
3D model (JSmol)	Interactive image
SMILES CN1CCC23CCCCC2C1Cc4ccc(O)cc34
InChI InChI=1S/C17H23NO/c1-18-9-8-17-7-3-2-4-14(17)16(18)10-12-5-6-13(19)11-15(12)17/h5-6,11,14,16,19H,2-4,7-10H2,1H3 Key:JAQUASYNZVUNQP-UHFFFAOYSA-N

Racemorphan

See also

References