List of combined sex-hormonal preparations

This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.

Androgens

Injection

Marketed

Veterinary

Marketed

Estrogens

Oral

Marketed

Injection

Marketed

  • Estradiol benzoate/estradiol phenylpropionate (Dimenformon Prolongatum)

Progestogens

Injection

Marketed

  • Progesterone/hydroxyprogesterone heptanoate/tocopherol (Tocogestan)

Androgens and estrogens

Oral

Marketed

  • Conjugated estrogens/methyltestosterone (Premarin with Methyltestosterone)
  • Dienestrol/methyltestosterone (Estan, Lucidon)
  • Esterified estrogens/methyltestosterone (Covaryx, Eemt, Essian, Estratest, Menogen, Syntest)
  • Ethinylestradiol/methyltestosterone (Mixogen)

Injection

Marketed

  • Estradiol/testosterone (Bothermon)
  • Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron)
  • Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Estandron P, Mixogen)
  • Estradiol benzoate/testosterone isobutyrate (Folivirin)
  • Estradiol cypionate/testosterone cypionate (Depo-Testadiol)
  • Estradiol hexahydrobenzoate/testosterone hexahydrobenzoate/hydroxyprogesterone caproate (Trinestril AP)
  • Estradiol valerate/prasterone enanthate (Binodian Depot, Cidodian Depot, Gynodian Depot, Supligol NF)
  • Estradiol valerate/testosterone enanthate (Despamen, Ditate-DS, Gravignost, Primodian Depot, Valertest)

Veterinary

Marketed

  • Diethylstilbestrol/methyltestosterone (Maxymin)
  • Diethylstilbestrol/testosterone (Rapigain)
  • Estradiol benzoate/estradiol enanthate/testosterone enanthate (Uni-Bol)
  • Estradiol benzoate/testosterone propionate (Component E-H, Implix BF, Progro H, Synovex H)
  • Ethinylestradiol/methyltestosterone (Taril)

Estrogens and progestogens

Oral

Marketed

In birth control pills:

  • Estradiol/nomegestrol acetate (Naemis, Zoely)
  • Estradiol valerate/cyproterone acetate (Femilar)
  • Estradiol valerate/dienogest (Natazia, Qlaira)
  • Ethinylestradiol/chlormadinone acetate (Belara)
  • Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
  • Ethinylestradiol/desogestrel (Desogen, Marvelon, Mercilon, Mircette, Novynette)
  • Ethinylestradiol/dienogest (Valette)
  • Ethinylestradiol/dimethisterone (Oracon)
  • Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
  • Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
  • Ethinylestradiol/etynodiol diacetate (Demulen)
  • Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
  • Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
  • Ethinylestradiol/levonorgestrel/bisglycinate
  • Ethinylestradiol/levonorgestrel/ferrous fumarate
  • Ethinylestradiol/lynestrenol (Lyndiol)
  • Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
  • Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
  • Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
  • Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
  • Ethinylestradiol/norethisterone acetate (FemHRT)
  • Ethinylestradiol/norethisterone acetate/ferrous fumarate
  • Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
  • Ethinylestradiol/norgestrel (Ovral)
  • Ethinylestradiol/norgestrienone (Miniplanor, Planor)
  • Ethinylestradiol/quingestanol acetate (Riglovis)
  • Mestranol/anagestone acetate (Neo-Novum)
  • Mestranol/chlormadinone acetate (C-Quens, Lutedion)
  • Mestranol/etynodiol diacetate (Ovulen)
  • Mestranol/lynestrenol (Lyndiol)
  • Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
  • Mestranol/noretynodrel (Enavid, Enovid)
  • Quinestrol/etynodiol diacetate (Soluna)
  • Quinestrol/levonorgestrel (Yuèkětíng, Àiyuè)
  • Quinestrol/norgestrel (Compound Norgestrel)
  • Quinestrol/quingestanol acetate (Unovis)

For menopausal hormone therapy:

  • Conjugated estrogens/medrogestone (Presomen)
  • Conjugated estrogens/medroxyprogesterone acetate (Prempro, Premphase)
  • Estradiol/cyproterone acetate (Climen)
  • Estradiol/drospirenone (Angeliq)
  • Estradiol/dydrogesterone (Femoston)
  • Estradiol/gestodene (Avaden, Avadene)
  • Estradiol/levonorgestrel
  • Estradiol/medroxyprogesterone acetate (Indivina, Tridestra)
  • Estradiol/norethisterone (Mimvey)
  • Estradiol/norethisterone acetate (Activella, Activelle, Cliane, Estalis, Eviana, Evorel, Kliogest, Novofem)
  • Estradiol/norgestimate (Prefest)
  • Estradiol/trimegestone (Lovelle, Totelle)
  • Estradiol valerate/cyproterone acetate (Climen 28)
  • Estradiol valerate/estriol/levonorgestrel (CycloÖstrogynal)
  • Estradiol valerate/levonorgestrel (Cyclo-Progynova N)
  • Estradiol valerate/medroxyprogesterone acetate (Dilena, Divina, Divitren, Farludiol, Indivina, Sisare)
  • Estradiol valerate/norethisterone (Climagest, Climesse)
  • Estradiol valerate/norethisterone acetate (Cliovelle, Norestin, Trisequens)
  • Estradiol valerate/norgestrel (Cyclacur, Cyclocur, Cyclo-Progynova, Postoval, Progyluton)

Not yet marketed

In birth control pills:

For menopausal hormone therapy:

Transdermal

Marketed

In contraceptive patches:

For menopausal hormone therapy:

Vaginal

Marketed

In contraceptive vaginal rings:

Injection

Marketed

In combined injectable contraceptives:

For menopausal hormone therapy, gynecological disorders, habitual abortion, and other indications:

Never marketed

In combined injectable contraceptives:

  • Estradiol undecylate/norethisterone enanthate
  • Estradiol valerate/gestonorone caproate (SH-834)
  • Estradiol valerate/methenmadinone acetate (Lutofollin)

Veterinary

Marketed

Androgens and progestogens

Veterinary

Marketed

  • Danazol/megestrol acetate (Dogalact)
  • Nandrolone decanoate/methandriol dipropionate (Filybol, Tribolin)
  • Nandrolone phenylpropionate/methandriol dipropionate (RWR)

Estrogens, progestogens, and androgens

Oral

Marketed

  • Methylestradiol/normethandrone (Ginecosid, Ginecoside, Mediol, Renodiol)

Injection

Marketed

  • Estradiol dibutyrate/testosterone caproate/hydroxyprogesterone heptanoate (Triormon Depositum)
  • Estradiol diundecylate/testosterone cyclohexylpropionate/hydroxyprogesterone heptanoate (Trioestrine Retard)

Never marketed

  • Estrapronicate/nandrolone decanoate/hydroxyprogesterone heptanoate (Trophobolene, Trophoboline)

Veterinary

Marketed

  • Estradiol/trenbolone acetate (Component, Compudose-G, Progro TE-H, Revalor, Synovex)
  • Estradiol benzoate/trenbolone acetate (Component TE-S, Synovex Choice, Synovex One, Synovex Plus)

Miscellaneous

Oral

Marketed

Mixed

Marketed

  • Goserelin/bicalutamide (ZolaCos CP)
  • Leuprorelin/norethisterone acetate (Lupaneta Pack)

See also

References

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