List of combined sex-hormonal preparations
This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.
Androgens
Injection
Marketed
- Testosterone propionate/testosterone enanthate (Testoviron depot)
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Sustanon 100)
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone decanoate (Sustanon 250)
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone caproate (Omnadren 250)
Veterinary
Marketed
Estrogens
Oral
Marketed
- Conjugated estriol (Emmenin, Progynon)
- Conjugated estrogens (Premarin)
- Esterified estrogens (Estratab, Menest)
- Estradiol/estrone/estriol (Hormonin)
- Ethinylestradiol/dienestrol (Foxinette)
Injection
Marketed
- Estradiol benzoate/estradiol phenylpropionate (Dimenformon Prolongatum)
Progestogens
Injection
Marketed
- Progesterone/hydroxyprogesterone heptanoate/tocopherol (Tocogestan)
Androgens and estrogens
Oral
Marketed
- Conjugated estrogens/methyltestosterone (Premarin with Methyltestosterone)
- Dienestrol/methyltestosterone (Estan, Lucidon)
- Esterified estrogens/methyltestosterone (Covaryx, Eemt, Essian, Estratest, Menogen, Syntest)
- Ethinylestradiol/methyltestosterone (Mixogen)
Injection
Marketed
- Estradiol/testosterone (Bothermon)
- Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron)
- Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Estandron P, Mixogen)
- Estradiol benzoate/testosterone isobutyrate (Folivirin)
- Estradiol cypionate/testosterone cypionate (Depo-Testadiol)
- Estradiol hexahydrobenzoate/testosterone hexahydrobenzoate/hydroxyprogesterone caproate (Trinestril AP)
- Estradiol valerate/prasterone enanthate (Binodian Depot, Cidodian Depot, Gynodian Depot, Supligol NF)
- Estradiol valerate/testosterone enanthate (Despamen, Ditate-DS, Gravignost, Primodian Depot, Valertest)
Veterinary
Marketed
- Diethylstilbestrol/methyltestosterone (Maxymin)
- Diethylstilbestrol/testosterone (Rapigain)
- Estradiol benzoate/estradiol enanthate/testosterone enanthate (Uni-Bol)
- Estradiol benzoate/testosterone propionate (Component E-H, Implix BF, Progro H, Synovex H)
- Ethinylestradiol/methyltestosterone (Taril)
Estrogens and progestogens
Oral
Marketed
- Estradiol/nomegestrol acetate (Naemis, Zoely)
- Estradiol valerate/cyproterone acetate (Femilar)
- Estradiol valerate/dienogest (Natazia, Qlaira)
- Ethinylestradiol/chlormadinone acetate (Belara)
- Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
- Ethinylestradiol/desogestrel (Desogen, Marvelon, Mercilon, Mircette, Novynette)
- Ethinylestradiol/dienogest (Valette)
- Ethinylestradiol/dimethisterone (Oracon)
- Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
- Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
- Ethinylestradiol/etynodiol diacetate (Demulen)
- Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
- Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
- Ethinylestradiol/levonorgestrel/bisglycinate
- Ethinylestradiol/levonorgestrel/ferrous fumarate
- Ethinylestradiol/lynestrenol (Lyndiol)
- Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
- Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
- Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
- Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
- Ethinylestradiol/norethisterone acetate (FemHRT)
- Ethinylestradiol/norethisterone acetate/ferrous fumarate
- Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
- Ethinylestradiol/norgestrel (Ovral)
- Ethinylestradiol/norgestrienone (Miniplanor, Planor)
- Ethinylestradiol/quingestanol acetate (Riglovis)
- Mestranol/anagestone acetate (Neo-Novum)
- Mestranol/chlormadinone acetate (C-Quens, Lutedion)
- Mestranol/etynodiol diacetate (Ovulen)
- Mestranol/lynestrenol (Lyndiol)
- Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
- Mestranol/noretynodrel (Enavid, Enovid)
- Quinestrol/etynodiol diacetate (Soluna)
- Quinestrol/levonorgestrel (Yuèkětíng, Àiyuè)
- Quinestrol/norgestrel (Compound Norgestrel)
- Quinestrol/quingestanol acetate (Unovis)
For menopausal hormone therapy:
- Conjugated estrogens/medrogestone (Presomen)
- Conjugated estrogens/medroxyprogesterone acetate (Prempro, Premphase)
- Estradiol/cyproterone acetate (Climen)
- Estradiol/drospirenone (Angeliq)
- Estradiol/dydrogesterone (Femoston)
- Estradiol/gestodene (Avaden, Avadene)
- Estradiol/levonorgestrel
- Estradiol/medroxyprogesterone acetate (Indivina, Tridestra)
- Estradiol/norethisterone (Mimvey)
- Estradiol/norethisterone acetate (Activella, Activelle, Cliane, Estalis, Eviana, Evorel, Kliogest, Novofem)
- Estradiol/norgestimate (Prefest)
- Estradiol/trimegestone (Lovelle, Totelle)
- Estradiol valerate/cyproterone acetate (Climen 28)
- Estradiol valerate/estriol/levonorgestrel (CycloÖstrogynal)
- Estradiol valerate/levonorgestrel (Cyclo-Progynova N)
- Estradiol valerate/medroxyprogesterone acetate (Dilena, Divina, Divitren, Farludiol, Indivina, Sisare)
- Estradiol valerate/norethisterone (Climagest, Climesse)
- Estradiol valerate/norethisterone acetate (Cliovelle, Norestin, Trisequens)
- Estradiol valerate/norgestrel (Cyclacur, Cyclocur, Cyclo-Progynova, Postoval, Progyluton)
Not yet marketed
- Estetrol/drospirenone (Estelle)
For menopausal hormone therapy:
- Estradiol/progesterone (TX-001HR, TX-12-001HR)
Transdermal
Marketed
- Ethinylestradiol/norelgestromin (Evra, Ortho Evra, Xulane)
For menopausal hormone therapy:
- Estradiol/levonorgestrel (Climara Pro)
- Estradiol/norethisterone acetate (Combipatch)
Vaginal
Marketed
In contraceptive vaginal rings:
- Ethinylestradiol/etonogestrel (Circlet, NuvaRing)
- Ethinylestradiol/segesterone acetate (Annovera)
Injection
Marketed
In combined injectable contraceptives:
- Estradiol/megestrol acetate (Chinese Injectable No. 2, Mego-E)
- Estradiol benzoate butyrate/algestone acetophenide (Redimen, Soluna, Unijab)
- Estradiol cypionate/medroxyprogesterone acetate (Cyclo-Provera, Cyclofem, Lunelle)
- Estradiol enanthate/algestone acetophenide (Anafertin, Deladroxate, Perlutan, Topasel, Yectames)
- Estradiol valerate/hydroxyprogesterone caproate (Chinese Injectable No. 1)
- Estradiol valerate/norethisterone enanthate (Mesigyna, Mesygest)
For menopausal hormone therapy, gynecological disorders, habitual abortion, and other indications:
- Estradiol/progesterone (Juvenum)
- Estradiol benzoate/hydroxyprogesterone caproate (Primosiston)
- Estradiol benzoate/progesterone (Duogynon)
- Estradiol dipropionate/hydroxyprogesterone caproate (EP Hormone Depot)
- Estradiol hemisuccinate/progesterone (Hosterona)
- Estradiol valerate/hydroxyprogesterone caproate (Gravibinan, Gravibinon)
- Estrone/progesterone (Synergon)
Never marketed
In combined injectable contraceptives:
- Estradiol undecylate/norethisterone enanthate
- Estradiol valerate/gestonorone caproate (SH-834)
- Estradiol valerate/methenmadinone acetate (Lutofollin)
Veterinary
Marketed
- Estradiol benzoate/progesterone (Component E-S, Implix BM, Synovex C, Synovex S)
- Estradiol valerate/norgestomet (Syncro-Mate-B)
Androgens and progestogens
Veterinary
Marketed
- Danazol/megestrol acetate (Dogalact)
- Nandrolone decanoate/methandriol dipropionate (Filybol, Tribolin)
- Nandrolone phenylpropionate/methandriol dipropionate (RWR)
Estrogens, progestogens, and androgens
Oral
Marketed
- Methylestradiol/normethandrone (Ginecosid, Ginecoside, Mediol, Renodiol)
Injection
Marketed
- Estradiol dibutyrate/testosterone caproate/hydroxyprogesterone heptanoate (Triormon Depositum)
- Estradiol diundecylate/testosterone cyclohexylpropionate/hydroxyprogesterone heptanoate (Trioestrine Retard)
Never marketed
- Estrapronicate/nandrolone decanoate/hydroxyprogesterone heptanoate (Trophobolene, Trophoboline)
Veterinary
Marketed
- Estradiol/trenbolone acetate (Component, Compudose-G, Progro TE-H, Revalor, Synovex)
- Estradiol benzoate/trenbolone acetate (Component TE-S, Synovex Choice, Synovex One, Synovex Plus)
Miscellaneous
Oral
Marketed
- Conjugated estrogens/bazedoxifene (Duavee)
Mixed
Marketed
- Goserelin/bicalutamide (ZolaCos CP)
- Leuprorelin/norethisterone acetate (Lupaneta Pack)
See also
References
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