DMPX
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Clinical data | |
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ATC code |
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Identifiers | |
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CAS Number | |
PubChem CID | |
ChemSpider | |
ECHA InfoCard |
100.162.258 |
Chemical and physical data | |
Formula | C10H10N4O2 |
Molar mass | 218.212 g/mol |
3D model (JSmol) | |
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DMPX (3,7-dimethyl-1-propargylxanthine) is a caffeine analog which displays affinity to A2 adenosine receptors, in contrast to the A1 subtype receptors.[1] DMPX had 28× and 15× higher potency than caffeine in blocking peripheral and central NECA-responses. The locomotor stimulation caused by DMPX (ED50 10 μmol/kg) was similarly higher than caffeine.[1]
See also
- DPCPX
- 8-PT
- CPX (8-CPT)
- 8-Chlorotheophylline
- Theophylline
References
- 1 2 3,7-Dimethyl-1-propargylxanthine: a potent and selective in vivo antagonist of adenosine analogs. Life Sci. 1988;43(21):1671-84. PMID 3193854
Receptor (ligands) |
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Transporter (blockers) |
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Enzyme (inhibitors) |
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See also: Receptor/signaling modulators |
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