Butaclamol
Butaclamol (AY-23,028) is a typical antipsychotic which was never marketed.[1] Sold as the hydrochloride salt for use in research, the compound acts as a dopamine receptor antagonist.[2]
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| Formula | C25H31NO |
| Molar mass | 361.529 g·mol−1 |
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Chemistry
pKa = 7.15 (uncorrected for ionic strength)[3]
References
- Buckingham, J (1985). Dictionary of organic compounds - Google Books. ISBN 9780412540905.
- http://www.sigmaaldrich.com/catalog/ProductDetail.do?D7=0&N5=SEARCH_CONCAT_PNO%7CBRAND_KEY&N4=D033%7CSIGMA&N25=0&QS=ON&F=SPEC
- F. A. Chrzanowski, B. A. McGrogan, B. E. Maryanoff (1985). "The pKa of butaclamol and the mode of butaclamol binding to central dopamine receptors." J. Med. Chem. 28 399-400.
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See also: Receptor/signaling modulators | |
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| Antidepressants (TCAs and TeCAs) |
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| Antihistamines |
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| Antipsychotics |
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